Application of Fluorine- And Nitrogen-Walk Approaches: Defining the Structural and Functional Diversity of 2-Phenylindole Class of Cannabinoid 1 Receptor Positive Allosteric Modulators

Sumanta Garai; Pushkar M. Kulkarni; Peter C. Schaffer; Luciana M. Leo; Asher L. Brandt; Ayat Zagzoog; Tallan Black; Xiaoyan Lin; Dow P. Hurst; David R. Janero; Mary E. Abood; Anaelle Zimmowitch; Alex Straiker; Roger G. Pertwee; Melanie Kelly; Anna Maria Szczesniak; Eileen M. Denovan-Wright; Ken Mackie; Andrea G. Hohmann; Patricia H. Reggio; Robert B. Laprairie; Ganesh A. Thakur

doi:10.1021/acs.jmedchem.9b01142

Application of Fluorine- And Nitrogen-Walk Approaches: Defining the Structural and Functional Diversity of 2-Phenylindole Class of Cannabinoid 1 Receptor Positive Allosteric Modulators

Sumanta Garai, Pushkar M. Kulkarni, Peter C. Schaffer, Luciana M. Leo, Asher L. Brandt, Ayat Zagzoog, Tallan Black, Xiaoyan Lin, Dow P. Hurst, David R. Janero, Mary E. Abood, Anaelle Zimmowitch, Alex Straiker, Roger G. Pertwee, Melanie Kelly, Anna Maria Szczesniak, Eileen M. Denovan-Wright, Ken Mackie, Andrea G. Hohmann, Patricia H. ReggioRobert B. Laprairie, Ganesh A. Thakur

科研成果: 期刊稿件 › 文章 › 同行评审

44 引用（Scopus）

源语言	英语
页（从-至）	542-568
页数	27
期刊	Journal of Medicinal Chemistry
卷	63
期	2
DOI	https://doi.org/10.1021/acs.jmedchem.9b01142
出版状态	已出版 - 1月 23 2020
已对外发布	是

!!!ASJC Scopus Subject Areas

分子药学
药物发现

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10.1021/acs.jmedchem.9b01142

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Garai, S., Kulkarni, P. M., Schaffer, P. C., Leo, L. M., Brandt, A. L., Zagzoog, A., Black, T., Lin, X., Hurst, D. P., Janero, D. R., Abood, M. E., Zimmowitch, A., Straiker, A., Pertwee, R. G., Kelly, M., Szczesniak, A. M., Denovan-Wright, E. M., Mackie, K., Hohmann, A. G., ... Thakur, G. A. (2020). Application of Fluorine- And Nitrogen-Walk Approaches: Defining the Structural and Functional Diversity of 2-Phenylindole Class of Cannabinoid 1 Receptor Positive Allosteric Modulators. Journal of Medicinal Chemistry, 63(2), 542-568. https://doi.org/10.1021/acs.jmedchem.9b01142

Application of Fluorine- And Nitrogen-Walk Approaches: Defining the Structural and Functional Diversity of 2-Phenylindole Class of Cannabinoid 1 Receptor Positive Allosteric Modulators. / Garai, Sumanta; Kulkarni, Pushkar M.; Schaffer, Peter C. 等.
在: Journal of Medicinal Chemistry, 卷 63, 号码 2, 23.01.2020, 页码 542-568.

科研成果: 期刊稿件 › 文章 › 同行评审

Garai, S, Kulkarni, PM, Schaffer, PC, Leo, LM, Brandt, AL, Zagzoog, A, Black, T, Lin, X, Hurst, DP, Janero, DR, Abood, ME, Zimmowitch, A, Straiker, A, Pertwee, RG, Kelly, M, Szczesniak, AM, Denovan-Wright, EM, Mackie, K, Hohmann, AG, Reggio, PH, Laprairie, RB & Thakur, GA 2020, 'Application of Fluorine- And Nitrogen-Walk Approaches: Defining the Structural and Functional Diversity of 2-Phenylindole Class of Cannabinoid 1 Receptor Positive Allosteric Modulators', Journal of Medicinal Chemistry, 卷 63, 号码 2, 页码 542-568. https://doi.org/10.1021/acs.jmedchem.9b01142

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title = "Application of Fluorine- And Nitrogen-Walk Approaches: Defining the Structural and Functional Diversity of 2-Phenylindole Class of Cannabinoid 1 Receptor Positive Allosteric Modulators",

author = "Sumanta Garai and Kulkarni, {Pushkar M.} and Schaffer, {Peter C.} and Leo, {Luciana M.} and Brandt, {Asher L.} and Ayat Zagzoog and Tallan Black and Xiaoyan Lin and Hurst, {Dow P.} and Janero, {David R.} and Abood, {Mary E.} and Anaelle Zimmowitch and Alex Straiker and Pertwee, {Roger G.} and Melanie Kelly and Szczesniak, {Anna Maria} and Denovan-Wright, {Eileen M.} and Ken Mackie and Hohmann, {Andrea G.} and Reggio, {Patricia H.} and Laprairie, {Robert B.} and Thakur, {Ganesh A.}",

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doi = "10.1021/acs.jmedchem.9b01142",

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AU - Schaffer, Peter C.

AU - Leo, Luciana M.

AU - Brandt, Asher L.

AU - Zagzoog, Ayat

AU - Black, Tallan

AU - Lin, Xiaoyan

AU - Hurst, Dow P.

AU - Janero, David R.

AU - Abood, Mary E.

AU - Zimmowitch, Anaelle

AU - Straiker, Alex

AU - Pertwee, Roger G.

AU - Kelly, Melanie

AU - Szczesniak, Anna Maria

AU - Denovan-Wright, Eileen M.

AU - Mackie, Ken

AU - Hohmann, Andrea G.

AU - Reggio, Patricia H.

AU - Laprairie, Robert B.

AU - Thakur, Ganesh A.

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Application of Fluorine- And Nitrogen-Walk Approaches: Defining the Structural and Functional Diversity of 2-Phenylindole Class of Cannabinoid 1 Receptor Positive Allosteric Modulators

!!!ASJC Scopus Subject Areas

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