Synthesis of 5′-Thymidine-Conjugated Formylphenylboronic Acids as Potential Lysine Targeting Iminoboronate Reversible Covalent Enzyme Probes

Alana M.M. Rangaswamy; Michael H.R. Beh; Ebrahim Soleimani; Steve Sequeira; Julie Cormier; Katherine N. Robertson; David L. Jakeman

doi:10.1021/acs.joc.2c01000

Synthesis of 5′-Thymidine-Conjugated Formylphenylboronic Acids as Potential Lysine Targeting Iminoboronate Reversible Covalent Enzyme Probes

Alana M.M. Rangaswamy, Michael H.R. Beh, Ebrahim Soleimani, Steve Sequeira, Julie Cormier, Katherine N. Robertson, David L. Jakeman

Economics, Econometrics and Finance

Research output: Contribution to journal › Article › peer-review

4 Citations (Scopus)

Original language	English
Pages (from-to)	13542-13555
Number of pages	14
Journal	Journal of Organic Chemistry
Volume	87
Issue number	21
DOIs	https://doi.org/10.1021/acs.joc.2c01000
Publication status	Published - Nov 4 2022

ASJC Scopus Subject Areas

Organic Chemistry

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10.1021/acs.joc.2c01000

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title = "Synthesis of 5′-Thymidine-Conjugated Formylphenylboronic Acids as Potential Lysine Targeting Iminoboronate Reversible Covalent Enzyme Probes",

author = "Rangaswamy, {Alana M.M.} and Beh, {Michael H.R.} and Ebrahim Soleimani and Steve Sequeira and Julie Cormier and Robertson, {Katherine N.} and Jakeman, {David L.}",

note = "Funding Information: We thank NSERC (RGPIN/03893, ALLRP/550135) and CIHR (153332) for financial support of this research. J.C. was an NSERC USRA recipient. Publisher Copyright: {\textcopyright} 2022 by the Author(s).",

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AU - Rangaswamy, Alana M.M.

AU - Beh, Michael H.R.

AU - Soleimani, Ebrahim

AU - Sequeira, Steve

AU - Cormier, Julie

AU - Robertson, Katherine N.

AU - Jakeman, David L.

N1 - Funding Information: We thank NSERC (RGPIN/03893, ALLRP/550135) and CIHR (153332) for financial support of this research. J.C. was an NSERC USRA recipient. Publisher Copyright: © 2022 by the Author(s).

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Synthesis of 5′-Thymidine-Conjugated Formylphenylboronic Acids as Potential Lysine Targeting Iminoboronate Reversible Covalent Enzyme Probes

ASJC Scopus Subject Areas

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