Novel Potent and Selective Agonists of the GPR55 Receptor Based on the 3-Benzylquinolin-2(1H)-One Scaffold

Costanza Ceni; Michael J. Benko; Kawthar A. Mohamed; Giulio Poli; Miriana Di Stefano; Tiziano Tuccinardi; Maria Digiacomo; Massimo Valoti; Robert B. Laprairie; Marco Macchia; Simone Bertini

doi:10.3390/ph15070768

Novel Potent and Selective Agonists of the GPR55 Receptor Based on the 3-Benzylquinolin-2(1H)-One Scaffold

Costanza Ceni, Michael J. Benko, Kawthar A. Mohamed, Giulio Poli, Miriana Di Stefano, Tiziano Tuccinardi, Maria Digiacomo, Massimo Valoti, Robert B. Laprairie, Marco Macchia, Simone Bertini

Research output: Contribution to journal › Article › peer-review

4 Citations (Scopus)

Original language	English
Article number	768
Journal	Pharmaceuticals
Volume	15
Issue number	7
DOIs	https://doi.org/10.3390/ph15070768
Publication status	Published - Jul 2022
Externally published	Yes

ASJC Scopus Subject Areas

Drug Discovery
Molecular Medicine
Pharmaceutical Science

Keywords

GPR55
GPR55 agonist
GPR55 modulator
benzylquinolin-2-one
p-ERK activation assay
quinolin-2-one

UN SDGs

This output contributes to the following UN Sustainable Development Goals (SDGs)

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10.3390/ph15070768

Cite this

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title = "Novel Potent and Selective Agonists of the GPR55 Receptor Based on the 3-Benzylquinolin-2(1H)-One Scaffold",

keywords = "GPR55, GPR55 agonist, GPR55 modulator, benzylquinolin-2-one, p-ERK activation assay, quinolin-2-one",

author = "Costanza Ceni and Benko, {Michael J.} and Mohamed, {Kawthar A.} and Giulio Poli and {Di Stefano}, Miriana and Tiziano Tuccinardi and Maria Digiacomo and Massimo Valoti and Laprairie, {Robert B.} and Marco Macchia and Simone Bertini",

note = "Publisher Copyright: {\textcopyright} 2022 by the authors. Licensee MDPI, Basel, Switzerland.",

year = "2022",

month = jul,

doi = "10.3390/ph15070768",

language = "English",

volume = "15",

journal = "Pharmaceuticals",

issn = "1424-8247",

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number = "7",

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TY - JOUR

T1 - Novel Potent and Selective Agonists of the GPR55 Receptor Based on the 3-Benzylquinolin-2(1H)-One Scaffold

AU - Ceni, Costanza

AU - Benko, Michael J.

AU - Mohamed, Kawthar A.

AU - Poli, Giulio

AU - Di Stefano, Miriana

AU - Tuccinardi, Tiziano

AU - Digiacomo, Maria

AU - Valoti, Massimo

AU - Laprairie, Robert B.

AU - Macchia, Marco

AU - Bertini, Simone

PY - 2022/7

Y1 - 2022/7

KW - GPR55

KW - GPR55 agonist

KW - GPR55 modulator

KW - benzylquinolin-2-one

KW - p-ERK activation assay

KW - quinolin-2-one

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U2 - 10.3390/ph15070768

DO - 10.3390/ph15070768

M3 - Article

AN - SCOPUS:85133025834

SN - 1424-8247

VL - 15

JO - Pharmaceuticals

JF - Pharmaceuticals

IS - 7

M1 - 768

ER -

Novel Potent and Selective Agonists of the GPR55 Receptor Based on the 3-Benzylquinolin-2(1H)-One Scaffold

ASJC Scopus Subject Areas

Keywords

UN SDGs

Access to Document

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