@article{52010f6d737f482986ead1ed5438e489,
title = "Mapping Cannabinoid 1 Receptor Allosteric Site(s): Critical Molecular Determinant and Signaling Profile of GAT100, a Novel, Potent, and Irreversibly Binding Probe",
keywords = "7-transmembrane receptor, Allosteric covalent probe, G protein-coupled receptors, allosteric site, biased signaling, binding domain, cannabinoid 1 receptor, cysteine, functional selectivity, homology modeling, isothiocyanate, ligand bias, ligand-binding motif, negative allosteric modulator, signal transduction, therapeutics discovery",
author = "Laprairie, {Robert B.} and Kulkarni, {Abhijit R.} and Kulkarni, {Pushkar M.} and Hurst, {Dow P.} and Diane Lynch and Reggio, {Patricia H.} and Janero, {David R.} and Pertwee, {Roger G.} and Stevenson, {Lesley A.} and Kelly, {Melanie E.M.} and Denovan-Wright, {Eileen M.} and Thakur, {Ganesh A.}",
note = "Publisher Copyright: {\textcopyright} 2016 American Chemical Society.",
year = "2016",
month = jun,
day = "15",
doi = "10.1021/acschemneuro.6b00041",
language = "English",
volume = "7",
pages = "776--798",
journal = "ACS Chemical Neuroscience",
issn = "1948-7193",
publisher = "American Chemical Society",
number = "6",
}